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- W2079551570 abstract "The water-soluble duocarmycin B1 prodrugs such as glycoside 3, phosphate 4 and carbamate 5 were synthesized for improving biological and pharmaceutical profiles of duocarmycin. Among these prodrugs, N-methylpiperazinylcarbamoyl derivative 5 exhibited potent antitumor activity against several human tumors in vivo." @default.
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- W2079551570 title "Synthesis and antitumor activity of water-soluble duocarmycin B1 prodrugs" @default.
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- W2079551570 doi "https://doi.org/10.1016/s0960-894x(99)00518-1" @default.
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