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- W2081943145 endingPage "1396" @default.
- W2081943145 startingPage "1387" @default.
- W2081943145 abstract "Background: μ-Opioid agonists have clinically useful effects and are used in a variety of acute and chronic pain conditions. However, repeated exposure to these drugs can lead to the development of physiologic dependence and, in some individuals, to opioid addiction. Objective: This review describes different rationales and modes of co-administration of opioid agonists and antagonists to increase and decrease the desired and undesired effects of the agonists. Methods: Publications in the English language were identified through a MEDLINE search and the bibliographies of identified articles were reviewed. Results/conclusions: The clinical indication is a crucial determinant of how opioid agonists and antagonists are co-administered and, in turn, the selection of mode of co-administration (i.e., sequential or simultaneous) determines the most appropriate type of antagonist, dosage and route of administration. However, because each clinical application has both benefits and limitations, it is suggested that co-administration parameters need to be adjusted to the specific requirements of individual patients." @default.
- W2081943145 created "2016-06-24" @default.
- W2081943145 creator A5032968625 @default.
- W2081943145 date "2008-05-12" @default.
- W2081943145 modified "2023-10-16" @default.
- W2081943145 title "Co-administration of opioid agonists and antagonists in addiction and pain medicine" @default.
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