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- W2085805439 endingPage "1952" @default.
- W2085805439 startingPage "1925" @default.
- W2085805439 abstract "The phenomenon of multidrug resistance (MDR) has attenuated the efficacy of anticancer drugs and the possibility of successful cancer chemotherapy. ATP-binding cassette (ABC) transporters play an essential role in mediating MDR in cancer cells by increasing efflux of drugs from cancer cells, hence reducing the intracellular accumulation of chemotherapeutic drugs. Interestingly, small-molecule tyrosine kinase inhibitors (TKIs), such as AST1306, lapatinib, linsitinib, masitinib, motesanib, nilotinib, telatinib and WHI-P154, have been found to have the capability to overcome anticancer drug resistance by inhibiting ABC transporters in recent years. This review will focus on some of the latest and clinical developments with ABC transporters, TKIs and anticancer drug resistance." @default.
- W2085805439 created "2016-06-24" @default.
- W2085805439 creator A5012459905 @default.
- W2085805439 creator A5016003061 @default.
- W2085805439 creator A5044867727 @default.
- W2085805439 creator A5055987305 @default.
- W2085805439 date "2014-09-29" @default.
- W2085805439 modified "2023-10-17" @default.
- W2085805439 title "Repositioning of Tyrosine Kinase Inhibitors as Antagonists of ATP-Binding Cassette Transporters in Anticancer Drug Resistance" @default.
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