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- W2090147678 abstract "A novel radioiodinated ligand of the butyrophenone type has been synthesized for the quantification and characterization of dopamine D2 receptors. This haloperidol-derived ligand, haloperidol-succinylglycyl[125I]iodotyrosine ([125I]HSGTI), binds rapidly (equilibrium is reached within 30 min, at 10 pM and 37 degrees C) and with high affinity (Kd = 0.3 nM) to bovine striatal membranes. Its pharmacology, determined by competitive displacement with dopaminergic and non-dopaminergic drugs, is characteristic of binding to dopamine D2 receptors." @default.
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- W2090147678 date "1987-11-30" @default.
- W2090147678 modified "2023-10-18" @default.
- W2090147678 title "Haloperidol-succinylglycyl[125I]iodotyrosine, a novel iodinated ligand for dopamine D2receptors" @default.
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- W2090147678 doi "https://doi.org/10.1016/0014-5793(87)80467-2" @default.
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