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- W2090148618 abstract "Amino acids 5 and 7, two potent and selective competitive GluR5 KA receptor antagonists, exhibited high GluR5 receptor affinity over other glutamate receptors. Their ester prodrugs 6 and 8 were orally active in three models of pain: reversal of formalin-induced paw licking, carrageenan-induced thermal hyperalgesia, and capsaicin-induced mechanical hyperalgesia." @default.
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- W2090148618 date "2005-05-21" @default.
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- W2090148618 title "Two Prodrugs of Potent and Selective GluR5 Kainate Receptor Antagonists Actives in Three Animal Models of Pain" @default.
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- W2090148618 doi "https://doi.org/10.1021/jm0491952" @default.
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