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- W2090876305 abstract "Efforts to modify the central proline portion of lead compound 4 lead to the discovery of novel prolylcarboxypeptidase (PrCP) inhibitors. Especially, replacement with alanine afforded compound 19 displaying more potent human and mouse PrCP inhibitory activity than 4 and an overall comparable profile." @default.
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- W2090876305 date "2012-02-01" @default.
- W2090876305 modified "2023-10-03" @default.
- W2090876305 title "Discovery of a new class of potent prolylcarboxypeptidase inhibitors derived from alanine" @default.
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- W2090876305 doi "https://doi.org/10.1016/j.bmcl.2011.12.064" @default.
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