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- W2091269938 abstract "[3H]verapamil binding to muscle tubule membrane has the following properties. KD = 27 ± 5 nM and maximum binding capacity Bmax = 50 ± 5 pmol/mg of protein. A 1 = 1 stoichiometry of binding was found for the ratio of [3H]verapamil versus [3H] nitrendipine binding sites. The dissociation constant found at equilibrium is near that determined from the ratio of the rate constants for association (k1) and dissociation (k−1). Antiarrhythmic drugs like D600, diltiazem and bepridil are competitive inhibitors of [3H]verapamil binding with KD values between 40 and 200 nM. Dihydropyridine analogs are apparent non competitive inhibitors of [3H]verapamil binding with half-maximum inhibition values (K0.5) between 1 and 5 nM." @default.
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- W2091269938 date "1984-01-01" @default.
- W2091269938 modified "2023-09-25" @default.
- W2091269938 title "[3H] verapamil binding sites in skeletal muscle tranverse tubule membranes" @default.
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- W2091269938 doi "https://doi.org/10.1016/0006-291x(84)91092-1" @default.
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