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- W2091448832 abstract "The synthesis, SAR and binding affinities of cannabinoid-1 receptor (CB1R) inverse agonists based on furo[2,3-b]pyridine scaffolds are described. Food intake, mechanism specific efficacy, pharmacokinetic, and metabolic evaluation of several of these compounds indicate that they are effective orally active modulators of CB1R." @default.
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- W2091448832 date "2010-02-01" @default.
- W2091448832 modified "2023-10-07" @default.
- W2091448832 title "Furo[2,3-b]pyridine-based cannabinoid-1 receptor inverse agonists: Synthesis and biological evaluation. Part 1" @default.
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- W2091448832 doi "https://doi.org/10.1016/j.bmcl.2009.12.065" @default.
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