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- W2094849619 abstract "Synthesis and biological evaluation of a series of 6-aminopyrazolyl-pyridine-3-carbonitriles as JAK2 kinase inhibitors was reported. Biochemical screening, followed by profile optimization, resulted in JAK2 inhibitors exhibiting good kinase selectivity, pharmacokinetic properties, physical properties and pharmacodynamic effects." @default.
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- W2094849619 date "2011-05-01" @default.
- W2094849619 modified "2023-10-10" @default.
- W2094849619 title "In vitro and in vivo evaluation of 6-aminopyrazolyl-pyridine-3-carbonitriles as JAK2 kinase inhibitors" @default.
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- W2094849619 doi "https://doi.org/10.1016/j.bmcl.2011.03.053" @default.
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