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- W2102016172 abstract "Chagas disease is caused by Trypanosoma cruzi, and is considered a public health problem. The current treatments for this disease are the synthetic drugs nifurtimox and benzonidazol, which are highly toxic. Pityrogramma calomelanos, a plant used in traditional medicine as an astringent, analgesic, anti-hemorrhagic, pectoral depurative, emmenagogue, anti-hypertensive, anti-pyretic and an anti-tussive was tested for antiepimastigote activity in vitro. An ethanol extract and hexane fraction of P. calomelanos was prepared and tested against T. cruzi (CL-B5 clone). The effective concentration capable of killing 50% of parasites (EC50) was 55.26 µg/mL and 73.57 µg/mL for the ethanol extract and hexane fraction, respectively. This is the first record of tripanocidal activity for P. calomelanos. Our results indicate that P. calomelanos could be a source of antiepimastigote natural products with only moderate toxicity toward healthy human cells." @default.
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- W2102016172 date "2012-07-01" @default.
- W2102016172 modified "2023-10-14" @default.
- W2102016172 title "Cytotoxic and Tripanocide Activities of Pityrogramma calomelanos (L.) Link" @default.
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- W2102016172 doi "https://doi.org/10.1640/0002-8444-102.3.198" @default.
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