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- W2107758429 endingPage "413" @default.
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- W2107758429 abstract "The signature action of aldosterone in the regulation of electrolyte and fluid balance is well established. However, the role of aldosterone as an important contributor to morbidity and mortality in heart failure has gained a heightened interest in recent years, but the mechanisms of this action are not well understood. Aldosterone is the principal physiological ligand for the mineralocorticoid receptor (MR), a ligand-activated transcription factor, that also binds to the physiological glucocorticoid, cortisol. Both classes of hormones bind with similar affinity to the MR, but the molecular basis of selective and tissue-specific effects of MR ligands is not yet fully documented. The structural and functional determinants of MR function are described and their significance is discussed." @default.
- W2107758429 created "2016-06-24" @default.
- W2107758429 creator A5046419066 @default.
- W2107758429 creator A5091861493 @default.
- W2107758429 date "2008-09-19" @default.
- W2107758429 modified "2023-10-15" @default.
- W2107758429 title "Structure–function relationships in the mineralocorticoid receptor" @default.
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- W2107758429 doi "https://doi.org/10.1677/jme-08-0093" @default.
- W2107758429 hasPubMedId "https://pubmed.ncbi.nlm.nih.gov/18805937" @default.
- W2107758429 hasPublicationYear "2008" @default.
- W2107758429 type Work @default.