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- W2111385909 endingPage "377" @default.
- W2111385909 startingPage "341" @default.
- W2111385909 abstract "Eukaryotic and prokaryotic organisms possess huge numbers of uncharacterized enzymes. Selective inhibitors offer powerful probes for assigning functions to enzymes in native biological systems. Here, we discuss how the chemical proteomic platform activity-based protein profiling (ABPP) can be implemented to discover selective and in vivo–active inhibitors for enzymes. We further describe how these inhibitors have been used to delineate the biochemical and cellular functions of enzymes, leading to the discovery of metabolic and signaling pathways that make important contributions to human physiology and disease. These studies demonstrate the value of selective chemical probes as drivers of biological inquiry." @default.
- W2111385909 created "2016-06-24" @default.
- W2111385909 creator A5002256644 @default.
- W2111385909 creator A5054637908 @default.
- W2111385909 date "2014-06-02" @default.
- W2111385909 modified "2023-10-11" @default.
- W2111385909 title "Enzyme Inhibitor Discovery by Activity-Based Protein Profiling" @default.
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