Matches in SemOpenAlex for { <https://semopenalex.org/work/W2112181688> ?p ?o ?g. }
- W2112181688 endingPage "132" @default.
- W2112181688 startingPage "108" @default.
- W2112181688 abstract "This review discusses anti-HIV natural products from several compound classes, including terpenoids, coumarins, alkaloids, polyphenols, tannins, and flavonoids. Natural products can provide novel anti-AIDS chemotherapeutic leads that are structurally unique or have new mechanisms of action. The drug discovery and development process proceeds from bioactivity-directed isolation and identification of a promising lead natural product, followed by rational design-based structural modification and structure-activity relationship analyses to optimize the lead compound as a drug candidate. This process is notably exemplified by the discovery of the modified betulinic acid derivative, DSB [PA-457], which is currently in Phase II clinical trial and is the first-in-class HIV maturation inhibitor (MI)." @default.
- W2112181688 created "2016-06-24" @default.
- W2112181688 creator A5000554610 @default.
- W2112181688 creator A5005512198 @default.
- W2112181688 creator A5043836895 @default.
- W2112181688 date "2006-01-01" @default.
- W2112181688 modified "2023-10-14" @default.
- W2112181688 title "New developments in natural products-based anti-AIDS research" @default.
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