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- W2112984940 endingPage "703" @default.
- W2112984940 startingPage "683" @default.
- W2112984940 abstract "Reversible histone methylation has emerged in the last few years as an important mechanism of epigenetic regulation. Histone methyltransferases and demethylases have been identified as contributing factors in the development of several diseases, especially cancer. Therefore, they have been postulated to be new drug targets with high therapeutic potential. Here, we review histone demethylases with a special focus on their potential role in oncology drug discovery. We present an overview over the different classes of enzymes, their biochemistry, selected data on their role in physiology and already available inhibitors." @default.
- W2112984940 created "2016-06-24" @default.
- W2112984940 creator A5016266091 @default.
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- W2112984940 creator A5074453653 @default.
- W2112984940 creator A5075157194 @default.
- W2112984940 creator A5085636203 @default.
- W2112984940 date "2012-08-07" @default.
- W2112984940 modified "2023-10-16" @default.
- W2112984940 title "The role of histone demethylases in cancer therapy" @default.
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