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- W2113041831 abstract "Ca1a2L analogues, having the central dipeptide a1a2 replaced by a sugar amino acid, were provided at the N-terminal end directly or via a spacer with a lipid. The inhibitory potency toward PGGT-1 of the set of lipophilic Ca1a2L analogues was improved in comparison with the original analogues, 1 and 2. The most potent inhibitors, 39 and 40, were found to inhibit PGGT-1 with an IC50-value of 12.7 and 12.3 μM, respectively, which is a 6-fold improvement over the corresponding analogue 1." @default.
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- W2113041831 date "2005-03-01" @default.
- W2113041831 modified "2023-09-27" @default.
- W2113041831 title "Synthesis and biological evaluation of lipophilic Ca1a2L analogues as potential bisubstrate inhibitors of protein:geranylgeranyl transferase-1" @default.
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- W2113041831 doi "https://doi.org/10.1016/j.bmc.2004.12.035" @default.
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