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- W2116480916 abstract "In-house screening of the Merck sample collection identified proline derived homophenylalanine 3 as a DPP-IV inhibitor with modest potency (DPP-IV IC50 = 1.9 μM). Optimization of 3 led to compound 37, which is among the most potent and selective DPP-IV inhibitors discovered to date." @default.
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- W2116480916 date "2004-10-01" @default.
- W2116480916 modified "2023-10-17" @default.
- W2116480916 title "Potent and selective proline derived dipeptidyl peptidase IV inhibitors" @default.
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- W2116480916 doi "https://doi.org/10.1016/j.bmcl.2004.07.056" @default.
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