Matches in SemOpenAlex for { <https://semopenalex.org/work/W2124804529> ?p ?o ?g. }
- W2124804529 abstract "Binding of salmon calcitonin to bovine hypothalamic membranes is enhanced about 25% by calcium with a half-maximal effect at 15 mM calcium. In contrast, membranes prepared from a cell line expressing a recombinant human calcitonin receptor show no effect of calcium under similar conditions. The hypothalamic calcitonin receptor solubilized with CHAPS detergent retains an apparent Kd of 0.3 nM for salmon calcitonin; however, binding of calcitonin to the detergent-solubilized receptor complex can be inhibited by divalent cations in order of potency Mn > Ca approximately Sr approximately Mg >> NaCl with Mn and Ca having apparent Ki's of 5 mM and 20 mM respectively. Dixon and Scatchard plots of Mn and Ca inhibition of binding to the soluble receptor complex suggest a noncompetitive mechanism of inhibition. Calcium also inhibits calcitonin binding to a detergent-solubilized recombinant human calcitonin receptor. Inhibition of calcitonin binding is observed using two independent methods for determining soluble receptor-hormone complex and inhibition is reversed by EDTA." @default.
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- W2124804529 date "1993-01-01" @default.
- W2124804529 modified "2023-10-18" @default.
- W2124804529 title "Modulation of Calcitonin Binding by Calcium: Differential Effects of Divalent Cations" @default.
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- W2124804529 doi "https://doi.org/10.3109/10799899309063271" @default.
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