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- W2126008082 abstract "Neuromuscular blockade following poisoning of the rat with DFP is shown to be rapidly antagonized by TMB-4 in vitro and in vivo . Concurrent study of the ChE activity following the addition of TMB-4 in vitro shows significant recovery of ChE activity of intact muscle after 10 minutes under the conditions used. Comparable results were obtained following TMB-4 treatment of sarin-poisoned rats.No reactivation of brain ChE activity was found following TMB-4 treatment, consistent with the apparent inability of quaternary compounds to penetrate the blood-brain barrier, and the potentiating action of atropine in promoting the chemotherapeutic effectiveness of TMB-4 shown previously." @default.
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- W2126008082 date "1960-12-01" @default.
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- W2126008082 title "Effects of 1,1'-trimethylene bis(4-formylpyridinium bromide) dioxime (TMB-4) on cholinesterase activity and neuromuscular block following poisoning with sarin and DEP." @default.
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