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- W2126943918 abstract "CP 96,345 is a nonpeptide high affinity antagonist of the substance P (NK1) receptor. The radiosynthesis of [11C]CP 96,345 suitable for Positron Emission Tomography (PET) applications is described. [11C]CP 96,345 was prepared by O-methylation of a desmethyl precursor via in situ generation of its phenolate salt. The in vivo tissue distribution of [11C]CP 96,345 in guinea pigs (n = 2) at 5 and 30 min was determined. Uptake was low in brain (approximately 0.04% dose/g) and highest (approximately 1-2% dose/g) in the spleen and lungs. The present findings indicate that the use of [11C]CP 96,345 in PET might be more applicable to the study of substance P receptors in peripheral tissues involved with inflammatory disease and arthritis." @default.
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- W2126943918 date "1993-05-01" @default.
- W2126943918 modified "2023-09-25" @default.
- W2126943918 title "Synthesis of a nonpeptide carbon-11 labeled substance P antagonist for PET studies" @default.
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- W2126943918 doi "https://doi.org/10.1016/0969-8051(93)90085-9" @default.
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