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- W2144174677 endingPage "978" @default.
- W2144174677 startingPage "959" @default.
- W2144174677 abstract "Background: The increasing number of kinases as potential drug targets, in combination with the need to screen large compound collections, demands the kinase assays to be homogeneous, non-radioactive, robust, sensitive, easy to miniaturize, and high-throughput. Objective: This review will focus on some of the chief biochemical and cellular kinase assay technologies and their applications in tyrosine kinase drug discovery. Methods: Recent literatures on these tyrosine kinase assay technologies are reviewed, each assay principle, advantages and drawbacks, as well as their potential utilities in tyrosine kinase drug discovery are discussed. Results/conclusion: There is no perfect assay yet; the choice of assay technology relies on the consideration of many factors including the intrinsic properties of the assay, intended application, cost, timeline, synergy with other in-house assay technologies and the expertise, familiarity and comfort level with certain technologies." @default.
- W2144174677 created "2016-06-24" @default.
- W2144174677 creator A5016271328 @default.
- W2144174677 creator A5041856800 @default.
- W2144174677 creator A5051085161 @default.
- W2144174677 creator A5084059598 @default.
- W2144174677 date "2008-07-16" @default.
- W2144174677 modified "2023-09-25" @default.
- W2144174677 title "Measuring the tyrosine kinase activity: a review of biochemical and cellular assay technologies" @default.
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- W2144174677 doi "https://doi.org/10.1517/17460441.3.8.959" @default.
- W2144174677 hasPubMedId "https://pubmed.ncbi.nlm.nih.gov/23484970" @default.
- W2144174677 hasPublicationYear "2008" @default.
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