Matches in SemOpenAlex for { <https://semopenalex.org/work/W2144940586> ?p ?o ?g. }
- W2144940586 endingPage "872" @default.
- W2144940586 startingPage "861" @default.
- W2144940586 abstract "Abstract The CXCR3 chemokine receptor was first discovered in 1996 and has been shown to play an important role in several diseases, most of which are related to inflammation. This review describes in detail the development of small CXCR3 ligands and their therapeutic potential. Classes of CXCR3 antagonists with strikingly variable core structures have emerged. Some of these compounds have confirmed the beneficial role of CXCR3 antagonism in animal models of disease. One of the compounds, AMG487, progressed to Phase II clinical trials but has been withdrawn because of lack of efficacy. New antagonist classes are being developed to reveal the full therapeutic potential of CXCR3." @default.
- W2144940586 created "2016-06-24" @default.
- W2144940586 creator A5016107952 @default.
- W2144940586 creator A5038589572 @default.
- W2144940586 creator A5044455499 @default.
- W2144940586 creator A5074907950 @default.
- W2144940586 creator A5087896916 @default.
- W2144940586 date "2008-06-05" @default.
- W2144940586 modified "2023-10-17" @default.
- W2144940586 title "Towards Small-Molecule CXCR3 Ligands with Clinical Potential" @default.
- W2144940586 cites W1480138027 @default.
- W2144940586 cites W1491294598 @default.
- W2144940586 cites W1511166699 @default.
- W2144940586 cites W1525077036 @default.
- W2144940586 cites W1565959221 @default.
- W2144940586 cites W1595430911 @default.
- W2144940586 cites W1622400382 @default.
- W2144940586 cites W169887259 @default.
- W2144940586 cites W1833104430 @default.
- W2144940586 cites W1837424662 @default.
- W2144940586 cites W1964408609 @default.
- W2144940586 cites W1966331477 @default.
- W2144940586 cites W1966447073 @default.
- W2144940586 cites W1968944419 @default.
- W2144940586 cites W1975684997 @default.
- W2144940586 cites W1981440980 @default.
- W2144940586 cites W1981644527 @default.
- W2144940586 cites W1988841714 @default.
- W2144940586 cites W1989035987 @default.
- W2144940586 cites W1989308725 @default.
- W2144940586 cites W1994060519 @default.
- W2144940586 cites W1994387916 @default.
- W2144940586 cites W1996183144 @default.
- W2144940586 cites W1997284331 @default.
- W2144940586 cites W1998605540 @default.
- W2144940586 cites W1999098706 @default.
- W2144940586 cites W2007184943 @default.
- W2144940586 cites W2009364468 @default.
- W2144940586 cites W2013888332 @default.
- W2144940586 cites W2014882192 @default.
- W2144940586 cites W2015863707 @default.
- W2144940586 cites W2017062485 @default.
- W2144940586 cites W2017958811 @default.
- W2144940586 cites W2023088800 @default.
- W2144940586 cites W2025930905 @default.
- W2144940586 cites W2026156526 @default.
- W2144940586 cites W2029824788 @default.
- W2144940586 cites W2035093405 @default.
- W2144940586 cites W2035581389 @default.
- W2144940586 cites W2038258688 @default.
- W2144940586 cites W2039137468 @default.
- W2144940586 cites W2044004371 @default.
- W2144940586 cites W2045281561 @default.
- W2144940586 cites W2046230726 @default.
- W2144940586 cites W2052379183 @default.
- W2144940586 cites W2053962612 @default.
- W2144940586 cites W2054065593 @default.
- W2144940586 cites W2057223279 @default.
- W2144940586 cites W2058902088 @default.
- W2144940586 cites W2066243575 @default.
- W2144940586 cites W2066301424 @default.
- W2144940586 cites W2069149379 @default.
- W2144940586 cites W2069150726 @default.
- W2144940586 cites W2069201165 @default.
- W2144940586 cites W2072178451 @default.
- W2144940586 cites W2073246701 @default.
- W2144940586 cites W2074422738 @default.
- W2144940586 cites W2081596482 @default.
- W2144940586 cites W2082042256 @default.
- W2144940586 cites W2086482022 @default.
- W2144940586 cites W2086642403 @default.
- W2144940586 cites W2091040274 @default.
- W2144940586 cites W2091586967 @default.
- W2144940586 cites W2094526634 @default.
- W2144940586 cites W2094850820 @default.
- W2144940586 cites W2096232692 @default.
- W2144940586 cites W2097813075 @default.
- W2144940586 cites W2104918497 @default.
- W2144940586 cites W2109062268 @default.
- W2144940586 cites W2109653742 @default.
- W2144940586 cites W2111732346 @default.
- W2144940586 cites W2115289037 @default.
- W2144940586 cites W2116493322 @default.
- W2144940586 cites W2117342688 @default.
- W2144940586 cites W2118064380 @default.
- W2144940586 cites W2119307374 @default.
- W2144940586 cites W2120446140 @default.
- W2144940586 cites W2124138140 @default.
- W2144940586 cites W2125852723 @default.
- W2144940586 cites W2129146910 @default.
- W2144940586 cites W2130858592 @default.
- W2144940586 cites W2131374005 @default.
- W2144940586 cites W2136376178 @default.
- W2144940586 cites W2139213208 @default.
- W2144940586 cites W2140478082 @default.
- W2144940586 cites W2140820106 @default.
- W2144940586 cites W2147064547 @default.
- W2144940586 cites W2149963584 @default.