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- W2148092969 abstract "In this study, we investigated the role of liver X receptor (LXR) in regulating cholesterol concentration in goose primary hepatocytes. Intracellular and extracellular cholesterol concentration, mRNA expression levels of genes related to phosphatidylinositol 3-kinase (PI3K) pathway, sterol regulatory element-binding protein 2 (SREBP-2), and 3-hydroxy-3-methylglutaryl-CoA reductase (HMGR) were measured in primary goose hepatocytes. We found that the intracellular cholesterol concentration showed an uptrend manner when the TO901317 concentration was under 1 μmol/L; compared with 1 μmol/L TO901317, 10 μmol/L TO901317 had an inhibiting effect (P<0.05). The regulation mode of SREBP-2 and HMGR gene expression is similar with that of intracellular cholesterol concentration. These data suggested that LXR activation may stimulate the cholesterol biosynthesis by activating expression of SREBP-2 and HMGR. Interestingly, the mRNA levels of genes related with PI3K pathway increased in the presence of TO901317, which suggested that LXR activation could promote PI3K signalling activity." @default.
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- W2148092969 date "2014-01-01" @default.
- W2148092969 modified "2023-09-25" @default.
- W2148092969 title "Effect of a Synthetic Liver X Receptor Agonist TO901317 on Cholesterol Concentration in Goose Primary Hepatocytes" @default.
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- W2148092969 doi "https://doi.org/10.4081/ijas.2014.2979" @default.
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