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- W2159156953 abstract "In whole segments of rabbit distal colon with mucosa removed, descending reflex relaxations of the circular muscle (descending inhibition) elicited by inflating (0.1-1 ml) an intraluminal balloon, were partially antagonized by 100 μM hexamethonium and the 5-HT3 receptor antagonist, ondansetron (3 μM), and abolished by 1 μM tetrodotoxin. The inhibitory effects of hexamethonium and ondansetron were additive. Conversely, hexamethonium (100 μM) and ondansetron (3 μM) failed to reduce electrically induced non-adrenergic non-cholinergic (NANC) relaxations of colonic circular muscle. It is concluded that interneuronally released acetylcholine and 5-hydroxytryptamine (5-HT) activate descending inhibitory pathways supplying the circular coat, via nicotinic and 5-HT3 receptors, respectively. This evidence suggests a functional involvement of 5-hydroxytryptaminergic transmission in the descending inhibition of rabbit colon." @default.
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- W2159156953 date "1995-11-01" @default.
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- W2159156953 title "5-HT3 receptor involvement in descending reflex relaxation in the rabbit isolated distal colon" @default.
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- W2159156953 doi "https://doi.org/10.1016/0014-2999(95)00565-3" @default.
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