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- W2168587099 abstract "The synthesis and SAR of a series of beta3 adrenoreceptor agonists based on a novel template derived from 4-aminomethylpiperidine coupled with a common pharmacophore, arylethylamine, is described. This combination led to the identification of human beta3 adrenoreceptor agonists with in vivo activity in a transgenic mouse model." @default.
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- W2168587099 date "2002-10-01" @default.
- W2168587099 modified "2023-09-25" @default.
- W2168587099 title "Novel substituted 4-aminomethylpiperidines as potent and selective human β3-agonists. Part 2: Arylethanolaminomethylpiperidines" @default.
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- W2168587099 doi "https://doi.org/10.1016/s0960-894x(02)00608-x" @default.
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