Matches in SemOpenAlex for { <https://semopenalex.org/work/W2170985017> ?p ?o ?g. }
- W2170985017 endingPage "295" @default.
- W2170985017 startingPage "269" @default.
- W2170985017 abstract "Peroxisome proliferator-activated receptors (PPARs) are ligand activated transcription factors that modulate target gene expression in response to endogenous and exogenous ligands. Ligands for the PPARs have been widely developed for the treatment of various diseases including dyslipidemias and diabetes. While targeting selective receptor activation is an established therapeutic approach for the treatment of various diseases, a variety of toxicities are known to occur in response to ligand administration. Whether PPAR ligands produce toxicity via a receptor-dependent and/or off-target-mediated mechanism(s) is not always known. Extrapolation of data derived from animal models and/or in vitro models, to humans, is also questionable. The different toxicities and mechanisms associated with administration of ligands for the three PPARs will be discussed, and important data gaps that could increase our current understanding of how PPAR ligands lead to toxicity will be highlighted." @default.
- W2170985017 created "2016-06-24" @default.
- W2170985017 creator A5040177618 @default.
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- W2170985017 creator A5073932699 @default.
- W2170985017 creator A5077633674 @default.
- W2170985017 creator A5081069263 @default.
- W2170985017 date "2005-12-01" @default.
- W2170985017 modified "2023-09-24" @default.
- W2170985017 title "The Toxicology of Ligands for Peroxisome Proliferator-Activated Receptors (PPAR)" @default.
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