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- W2171396119 abstract "The inside cover picture shows two inhibitors of cathepsin (cat) L and B that are structural analogues but have different potency and selectivity against the two targets. Analysis of similarity and potency or selectivity distributions in molecular networks elucidates structure–activity and structure–selectivity relationships and identifies compounds forming activity and selectivity cliffs. For more details, see the Full Paper by J. Bajorath et al. on p. 1864 ff." @default.
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- W2171396119 date "2009-11-02" @default.
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- W2171396119 title "Inside Cover: From Structure-Activity to Structure-Selectivity Relationships: Quantitative Assessment, Selectivity Cliffs, and Key Compounds (ChemMedChem 11/2009)" @default.
- W2171396119 doi "https://doi.org/10.1002/cmdc.200990052" @default.
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