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- W2174260023 abstract "A series of anilino(imidazoquinoxaline) analogues bearing solubilizing side chains at the 6- and 7-positions of the fused phenyl ring has been prepared and evaluated for inhibition against Lck enzyme and of T-cell proliferation. Significant improvement of the cellular activity was achieved over the initial lead, compound 2." @default.
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- W2174260023 date "2002-11-01" @default.
- W2174260023 modified "2023-09-27" @default.
- W2174260023 title "Synthesis and SAR of novel imidazoquinoxaline-Based Lck inhibitors: improvement of cell potency" @default.
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- W2174260023 doi "https://doi.org/10.1016/s0960-894x(02)00677-7" @default.
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