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- W2174366973 endingPage "2012" @default.
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- W2174366973 abstract "1-Phenyl-8-azabicyclo[3.2.1]octane ethers are NK(1) receptor antagonists. Substitution at the 6-exo-position led to high affinity NK(1) antagonists with a prolonged duration of action in vivo. Incorporation of an alpha-methyl substituent in the pendent benzyl ether side chain gave compounds with increased selectivity over the hERG channel." @default.
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- W2174366973 date "2006-04-01" @default.
- W2174366973 modified "2023-10-18" @default.
- W2174366973 title "1-Phenyl-8-azabicyclo[3.2.1]octane ethers: A novel series of neurokinin (NK1) antagonists" @default.
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- W2174366973 doi "https://doi.org/10.1016/j.bmcl.2005.12.069" @default.
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