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- W2177531701 abstract "The discovery of N-substituted-pyridoindolines and their binding affinities at the 5-HT2A, 5-HT2C and D2 receptors, and in vivo efficacy as 5-HT2A antagonists is described. The structure–activity relationship of a series of core tetracyclic derivatives with varying butyrophenone sidechains is also discussed. This study has led to the identification of potent, orally bioavailable 5-HT2A/D2 receptor dual antagonists as potential atypical antipsychotics." @default.
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- W2177531701 date "2003-02-01" @default.
- W2177531701 modified "2023-09-27" @default.
- W2177531701 title "Novel, highly potent, selective 5-HT2A/D2 receptor antagonists as potential atypical antipsychotics" @default.
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- W2177531701 doi "https://doi.org/10.1016/s0960-894x(02)01028-4" @default.
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