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- W2186641987 abstract "Etoricoxib, a widely prescribed anti-inflammatory and analgesic drug belongs to class II under BCS and exhibit low and variable oral bioavailability due to its poor aqueous solubility. It is practically insoluble in water and aqueous fluids. As such its oral absorption is dissolution rate limited and it requires enhancement in solubility and dissolution rate for increasing its oral bioavailability. The objective of the present study is to enhance the solubility and dissolution rate of etoricoxib employing β-cyclodextrin (βCD) and two surfactants (SLS and Tween 80) alone and in combination. The individual main effects and combined (interaction) effects of βcyclodextrin and surfactants on the solubility and dissolution rate of etoricoxib were evaluated in a series of 2 2" @default.
- W2186641987 created "2016-06-24" @default.
- W2186641987 creator A5064132364 @default.
- W2186641987 date "2012-01-01" @default.
- W2186641987 modified "2023-09-27" @default.
- W2186641987 title "A FACTORIAL STUDY ON ENHANCEMENT OF SOLUBILITY AND DISSOLUTION RATE OF ETORICOXIB EMPLOYING β-CYCLODEXTRIN AND SURFACTANTS" @default.
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- W2186641987 hasPublicationYear "2012" @default.
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