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- W2228239295 startingPage "7" @default.
- W2228239295 abstract "Tau deposition is one of the neuropathological hallmarks in Alzheimer's disease as well as in other neurodegenerative disorders called tauopathies. Recent efforts to develop selective tau radiopharmaceuticals have allowed the visualization of tau deposits in vivo. In vivo tau imaging allows the assessment of the regional distribution of tau deposits in a single human subject over time for determining the pathophysiology of tau accumulation in aging and neurodegenerative conditions as well as for application in drug discovery of anti-dementia drugs as surrogate markers. However, tau deposits show complicated characteristics because of different isoform composition, histopathology, and ultrastructure in various neurodegenerative conditions. In addition, since tau radiopharmaceuticals possess different chemotype classes, they may show different binding characteristics with heterogeneous tau deposits. In this review, we describe the characteristics of tau deposits and their ligands that have β-sheet binding properties, and the status of tau imaging in clinical studies." @default.
- W2228239295 created "2016-06-24" @default.
- W2228239295 creator A5015270336 @default.
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- W2228239295 creator A5028540036 @default.
- W2228239295 creator A5035847289 @default.
- W2228239295 creator A5042373488 @default.
- W2228239295 creator A5063415107 @default.
- W2228239295 creator A5065225018 @default.
- W2228239295 date "2016-01-06" @default.
- W2228239295 modified "2023-10-07" @default.
- W2228239295 title "Characteristics of Tau and Its Ligands in PET Imaging" @default.
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