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- W2234664680 endingPage "97" @default.
- W2234664680 startingPage "67" @default.
- W2234664680 abstract "Drug transporters play indispensable roles in the disposition of drugs in the body; e.g., in hepatic and renal eliminations, intestinal absorption, and in transport across active barriers, and consequently, in the response to drugs. Importance of the solute carrier family, such as OATP/SLCO, OCT/SLC22, OAT/SLC22, and MATE/SLC47, and the ATP-binding cassette transporters, such as P-glycoprotein/ABCB1, MRPs/ABCC, and BCRP/ABCG2, are well recognized in drug discovery and clinical situations. To date, it is however a great challenge to identify in vivo probe substrates and inhibitors applicable for investigating the impact of drug transporters in humans. This chapter has summarized the relevant clinical drug–drug interaction and pharmagenomic studies on drug transporters in humans, as well as some in vitro studies on transporters, in order to suggest applicable probe substrates and inhibitors for drug transporters. In addition to the drugs at the market, some endogenous and food-derived metabolites are probes for drug transporters. This chapter also highlights the impact of drug transporters on such compounds." @default.
- W2234664680 created "2016-06-24" @default.
- W2234664680 creator A5027984186 @default.
- W2234664680 creator A5061014418 @default.
- W2234664680 creator A5088638080 @default.
- W2234664680 date "2013-01-01" @default.
- W2234664680 modified "2023-10-16" @default.
- W2234664680 title "In Vivo Characterization of Interactions on Transporters" @default.
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