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- W2245285550 abstract "Objective:To study the effects of polyamine analogue BENS [N1, N11-bis(ethyl) norspermine] on proliferation and apoptosis of melanoma cell line B16-F1. Methods:MTT assay was used to assess the viability of cells. The apoptotic rate was determined by flow cytometry. The change in cell membrane potential was measured by fluorescence staining. Cell apoptosis was evaluated by DNA fragmentation assays. The levels of apoptosis-related proteins were measured by Western blotting. Results:The polyamine analogue BENS markedly inhibited the proliferation of B16-F1 cells in a dose-dependent manner. BENS treatment resulted in DNA fragmentation and appearance of typical sub-G1 peak which was accompanied by apoptosis-related changes such as decrease in the mitochondrial membrane potential, release of cytochrome C from mitochondria to cytosol, and translocation of Bax from cytosol to mitochondria. Conclusion:The polyamine analogue BENS inhibits growth and induces apoptosis of melanoma B16-F1 cells. It indicates that BENS has potential values in clinical cancer therapy." @default.
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- W2245285550 date "2009-01-01" @default.
- W2245285550 modified "2023-09-22" @default.
- W2245285550 title "Effect of polyamine analogue BENS on proliferation of melanoma B16-F1 cells" @default.
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