Matches in SemOpenAlex for { <https://semopenalex.org/work/W22474514> ?p ?o ?g. }
- W22474514 endingPage "295" @default.
- W22474514 startingPage "267" @default.
- W22474514 abstract "β-Arrestins 1 and 2 are ubiquitously expressed proteins that play a dual role in G protein-coupled receptor (GPCR) signaling. On the one hand, arrestins are central to the termination of G protein-mediated receptor signaling and subsequent clathrin-dependent internalization. On the other hand, these proteins act as molecular scaffolds for G protein-independent GPCR signaling. This review provides an overview of how these dual functions of arrestins contribute to the biological outcomes associated to the activation of different brain GPCR. It also explores recent evidence suggesting how the dual function of arrestins can lead to the development of more selective pharmacological approaches for the treatment of central nervous system disorders such as chronic pain, bipolar disorder, major depression, and schizophrenia. Development of such approaches may lead to new drugs having better clinical efficacy and lesser side effects." @default.
- W22474514 created "2016-06-24" @default.
- W22474514 creator A5058693559 @default.
- W22474514 creator A5089009747 @default.
- W22474514 date "2013-01-01" @default.
- W22474514 modified "2023-09-27" @default.
- W22474514 title "β-Arrestins in the Central Nervous System" @default.
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