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- W2253808368 abstract "A bacterial defense mechanism Polymyxins are antibiotics that disrupt the bacterial cell membrane and are used to treat multidrug-resistant infections. A bacterial enzyme called ArnT can mediate resistance to polymyxins by transferring a sugar group from a lipid carrier to lipid A, a component of the bacterial outer membrane. Petrou et al. described structures of ArnT alone and in complex with a lipid carrier and identified a cavity where lipid A probably binds. Insights into the enzyme mechanism could be exploited to design drugs that combat polymyxin resistance. Science , this issue p. 608" @default.
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- W2253808368 date "2016-02-05" @default.
- W2253808368 modified "2023-10-17" @default.
- W2253808368 title "Structures of aminoarabinose transferase ArnT suggest a molecular basis for lipid A glycosylation" @default.
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- W2253808368 doi "https://doi.org/10.1126/science.aad1172" @default.
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