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- W2255827635 abstract "本文通过简单可行的方法合成了一个4-苯胺喹唑啉衍生物1,并通过分子对接的方法探讨了其JAK3抑制活性的分子作用机制。结果表明,化合物1与JAK3蛋白中ATP活性位点的关键氨基酸残基有一系列的相互作用,对JAK3蛋白的亲和力高于JANEX-1和Tasocitinib,呈现较强的JAK3抑制活性。" @default.
- W2255827635 created "2016-06-24" @default.
- W2255827635 creator A5031303874 @default.
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- W2255827635 date "2011-03-15" @default.
- W2255827635 modified "2023-09-25" @default.
- W2255827635 title "Synthesis and molecular docking study of (E)-4-(6,7-dimethoxyquinazolin-4-ylamino)phenyl-3-(4-chlorophenyl)acrylate as a JAK3 inhibitor" @default.
- W2255827635 doi "https://doi.org/10.5246/jcps.2011.02.014" @default.
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