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- W2316483451 abstract "The incidence of cutaneous melanoma isrisingmorerapidlythanthatforanyotherma-lignant tumor. If distant metastases occur, theannual survival falls below 20% [Keilholz etal. 2001]. Temozolomide (TMZ) and dacar-bazine (DTIC) as monochemotherapy, areconsidered the standard therapy for metasta-sized and surgically unresectable melanoma.An approximately 15% objective responseratecanbeachievedwithDTIC[Serroneetal.2000].The chemotherapeutic agents TMZ andDTIC are pro-drugs of the cytotoxic agent5-(3-methyltriazen-1-yl)imidazole-4-carbox-amide (MTIC) [Serrone et al. 2000]. MTICpossesses alkylating activity and generatesmethyl-DNA-adducts. The most crucialmethyl-DNA-adductfortheefficacyofTMZ/DTICtreatmentisO" @default.
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- W2316483451 date "2009-01-01" @default.
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- W2316483451 title "Modulation of the efficacy of temozolomide and dacarbazine melanoma treatment by DNA-repair factors in vivo and in vitro" @default.
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- W2316483451 doi "https://doi.org/10.5414/cpp47033" @default.
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