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- W2317354920 abstract "The mouse thymoma R1.1 cell line expresses a κ opioid receptor that is negatively coupled to adenylyl cyclase through a pertussis toxin-sensitive G i protein. This study addressed whether chronic exposure of R1.1 cells to the κ agonist U50,488 would alter the receptor binding properties or opioid-induced inhibition of adenylyl cyclase activity. Culturing R1.1 cells in the presence of U50,488 for 3 hr and longer produced a time- and concentration-dependent decrease in the binding of the κ-selective ligand [ 3 U]69,593 to membranes prepared from these cells. Unlike the decrease in receptor binding, opioid imbibition of adenylyl cyclase activity was not altered by culturing cells in the presence of U50,488" @default.
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- W2317354920 date "1994-02-01" @default.
- W2317354920 modified "2023-09-23" @default.
- W2317354920 title "Chronic opioid treatment of R1.1 cells results in the downregulation of the kappa opioid receptor without desensitization of adenylyl cyclase activity" @default.
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- W2317354920 doi "https://doi.org/10.1016/0167-0115(94)90301-8" @default.
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