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- W2321837669 abstract "Resume La dapsone, decouverte en 1908, appartient a la classe des sulfones. C'est le traitement de reference de la lepre depuis les annees 1940 et ses indications se sont ensuite etendues a d'autres infections et a des dermatoses inflammatoires. Ces indications reposent sur ses effets antibiotiques (lepre, pneumocystose…) et immunomodulateurs (dermatoses bulleuses auto-immunes, dermatoses neutrophiliques…). Sa biodisponibilite et sa demi-vie longue permettent une prise orale uniquotidienne. La dapsone est metabolisee par deux voies enzymatiques : N-acetylation et N-hydroxylation. Ses metabolites N-hydroxyles sont responsables de ses effets indesirables dose-dependants : hemolyse et methemoglobinemie. La dapsone presente egalement des effets indesirables idiosyncrasiques (agranulocytose, syndrome d'hypersensibilite)." @default.
- W2321837669 created "2016-06-24" @default.
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- W2321837669 date "2006-01-01" @default.
- W2321837669 modified "2023-09-26" @default.
- W2321837669 title "Dapsone (Disulone®) en dermatologie" @default.
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