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- W2327014777 abstract "A series consisting of ianthelliformisamimes A, B, and C as well as its synthetic analogues was prepared in high chemical yield, from 27 to 91%, using peptide coupling as the key step, and the compounds were evaluated for their in vitro antibiotic enhancer properties against resistant Gram-negative bacteria and clinical isolates. The mechanism of action of one of these derivatives against Pseudomonas aeruginosa when combined with doxycycline was precisely evaluated utilizing bioluminescence to measure ATP efflux and fluorescence to evaluate membrane depolarization." @default.
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- W2327014777 date "2014-05-13" @default.
- W2327014777 modified "2023-10-18" @default.
- W2327014777 title "New Ianthelliformisamine Derivatives as Antibiotic Enhancers against Resistant Gram-Negative Bacteria" @default.
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- W2327014777 doi "https://doi.org/10.1021/jm500194e" @default.
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