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- W23271723 abstract "Publisher Summary This chapter discusses the key biological and structural features of HIV protease (HIV PR) that define its usefulness as an antiviral target. HIV proteases have proven to be valuable instructional targets for the design of mechanism- and structure-based drugs, and for providing novel strategies for designing antiviral therapeutics. The introduction of PR inhibitors to the armamentarium of AIDS drugs has had a profoundly successful impact on the AIDS community where these drugs are prolonging life and providing new hope for the long-term maintenance of relatively good health until such time as a more effective cure or vaccine becomes available. The chapter presents a brief review as well as an update on efforts to discover and design inhibitors of HIV PR inhibitors. The problem of drug resistance to HIV PR inhibitors is discussed with an emphasis on viral strategies for resistance and on implications for future drug discovery efforts in this area." @default.
- W23271723 created "2016-06-24" @default.
- W23271723 creator A5037802350 @default.
- W23271723 creator A5045668817 @default.
- W23271723 date "1999-01-01" @default.
- W23271723 modified "2023-10-16" @default.
- W23271723 title "HIV Protease as a Target for the Design of Antiviral Agents for AIDS" @default.
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