Matches in SemOpenAlex for { <https://semopenalex.org/work/W2338275023> ?p ?o ?g. }
- W2338275023 abstract "Abstract DNA methylation and modifications of histones, such as reversible acetylation and methylation on lysine residues, are very important for epigenetic regulation. Methyl-lysine binding proteins recognize distinct lysine residues within proteins and they distinguish between different levels of methylation. Signaling events and biological outcome of histone methylation are mediated by methyl-lysine binding proteins which are also referred to as readers of the epigenetic code. The involvement of methyl-lysine readers in different diseases makes them highly promising drug targets that might result in novel therapeutic strategies in the future. In this chapter, early drug discovery approaches in this field are introduced and small-molecule inhibitors of the interaction of reader proteins and their histone-binding partners are presented. Furthermore, this chapter reviews the literature on reader proteins that are reported to function as oncoproteins and thus display potential drug targets." @default.
- W2338275023 created "2016-06-24" @default.
- W2338275023 creator A5008197229 @default.
- W2338275023 creator A5016266091 @default.
- W2338275023 creator A5089212888 @default.
- W2338275023 creator A5090341188 @default.
- W2338275023 date "2016-01-01" @default.
- W2338275023 modified "2023-10-17" @default.
- W2338275023 title "Epigenetic Readers Interpreting the Lysine Methylome—Biological Roles and Drug Discovery" @default.
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