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- W2350917246 abstract "Objective The hypotension of AT1 receptor knockout mice(AT1A-/-)can be,at least in part,explained by AT1 receptor deficiency.However,whether there is mechanism beyond AT1 receptor is not known.Our previous study showed negatively interaction between D5 dopamine receptor and AT1 receptor.Based on above-mentioned evidences,we hypothesize that D5 receptor is involved in the pathogenesis of hypotension of AT1A-/-mice.Methods Blood pressure,urine natriuretic excretion,renal D5 receptor expression were investigated in AT1A-/-mice and their control(AT1A+/+)mice.Furthermore,the mutual interaction between AT1 receptor and D5 receptor was also investigated in renal proximal tubule(RPT)cells from Wistar-Kyoto(WKY)rats and D5 receptor transfected HEK293 cells.Results As compared with AT1A+/+ mice,AT1A-/-mice on low-salt diet had lower blood pressure,higher renal D5 receptor expression.Stimulation of AT1 receptor with angiotensin Ⅱ decreased D5 receptors in WKY cells.Moreover,stimulation of D5 receptor also decreased AT1 receptor expression in D5 receptor transfected HEK293 cells.Conclusion Higher renal D5 receptor expression might be involved in the pathogenesis of hypotension of AT1A-/-mice." @default.
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- W2350917246 date "2007-01-01" @default.
- W2350917246 modified "2023-09-25" @default.
- W2350917246 title "Role of D_5 dopamine Receptors in Hypotension of AT1 Receptor Knock-out Mice" @default.
- W2350917246 hasPublicationYear "2007" @default.
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