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- W2360193090 abstract "AIM: To demonstrate the effect of mitochondrial ATP-sensitive potassium channel opener,Diazoxide,on glutamate uptake activity of astrocyte. METHODS: Primary astrocytic cultures were prepared from cerebral cortices of rats within 3 days old.Glutamate uptake activity of astrocytes was measured using isotopic techniques to detect intracellular -labeled D,L-glutamate concentration.RESULTS: Diazoxide increased -glutamate uptake in a concentration-dependent manner,and could significantly reverse MPP~+-induced glutamate uptake inhibition.The above effects of Diazoxide were blocked by 5-hydroxydecanoate,a selective mitochondrial ATP-sensitive potassium channel blocker.CONCLUSION: Diazoxide increase the activity of glutamate transporters in astrocytes by opening mitochondrial ATP-sensitive potassium channel." @default.
- W2360193090 created "2016-06-24" @default.
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- W2360193090 date "2006-01-01" @default.
- W2360193090 modified "2023-09-28" @default.
- W2360193090 title "Diazoxide increases glutamate uptake by astrocytes via activating mitochondrial ATP-sensitive potassium channels" @default.
- W2360193090 hasPublicationYear "2006" @default.
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