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- W2363301116 abstract "Objective To investigate whether tamoxifen reverses the resistance to VP16 mediated by breast cancer resistance protein.Methods Toxicity of tamoxifen,VP16 and VP16 combined with tamoxifen in JAR and JAR/VP16 cell line was detected by MTT.Intracell fluorescence intensity of hochest 33342 and PI was accessed by flow cytometery.Expressions of BCRP mRNA and protein in JAR and JAR/VP16 cell line were detected by RT-PCR and Western blot.Results The expression of BCRP was upregulated in JAR/VP16 cell line.Effect of VP16 could be enhanced by tamoxifen. Cell inhibition ratio was significantly increased when VP16 combined with tamoxifen(P0.05).Expression of BCRP could be downregulated by tamoxifen. Conclusion Overexpression of BCRP results in the resistance of JAR/VP16 cell line to VP16.Tamoxifen can reverse the resistance via downregulating BCRP and inhibiting the function of BCRP." @default.
- W2363301116 created "2016-06-24" @default.
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- W2363301116 date "2007-01-01" @default.
- W2363301116 modified "2023-09-24" @default.
- W2363301116 title "Tamoxifen reverses the resistance to VP16 in breast cancer resistance protein overexpression cell line JAR/VP16 to VP16" @default.
- W2363301116 hasPublicationYear "2007" @default.
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