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- W2379075093 abstract "Objective: This study was designed to examine the interaction between rocuronium and vecuronium or atracurium on adult-and embryonic-muscular nicotinic acetylcholine receptors with whole cell clamp patch. Methods: The adult-and embryonic-nicotinic acetylcholine receptors were heterologously expressed in HEK293 cells. Peak currents were recorded in HEK293 cells treated by rocuronium,vecuronium,atracurium individually using whole cell patch clamp technique. Drug combinations containing equipotent concentrations of rocuronium and vecuronium or rocuronium and atracurium were tested and dose-response curves were determined. Results: All compounds tested alone and in combination produced rapid and readily reversible,concentration-dependent inhibition. Two agents with similar or dissimilar structure were combined in equipotent concentrations. Isobolographic analysis indicated additive interaction for combination of rocuronium and vecuronium on embryonic receptor and synergistic interaction on adult receptor,whereas isobolographic analysis of combination of rocuronium and atracurium indicated synergistic interaction on both adult-and embryonic-nicotinic acetylcholine receptors. Conclusion: The interactions of combination of muscle relaxants with dissimilar structure,rocuronium and atracurium were synergistic to both adult-and embryonic-nicotinic acetylcholine receptors and with similar structure,rocuronium and vecuronium were synergistic to adult-nicotinic acetylcholine receptors and additive to embryonic-nicotinic acetylcholine receptors." @default.
- W2379075093 created "2016-06-24" @default.
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- W2379075093 date "2008-01-01" @default.
- W2379075093 modified "2023-09-28" @default.
- W2379075093 title "Effects of Rocuronium Combined with Vecuronium and Atracurium on Adult-and Embryonic-Muscular Nicotinic Acetylcholine Receptors" @default.
- W2379075093 hasPublicationYear "2008" @default.
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