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- W2382173 endingPage "135" @default.
- W2382173 startingPage "101" @default.
- W2382173 abstract "Drugs that are known to activate or block dopamine receptors are widely used for the treatment of a number of severe diseases. In most cases, dopaminergic drugs preferentially interact with the subtypes of the D2 family (D2, D3, D4). However, only minor selectivity has been observed between D2, D3, and D4. Nevertheless, in recent years D3 and D4 subtype-selective agonists, partial agonists, and antagonist have been developed. The most interesting structural features required for high selectivity and affinity are presented as well as structure–activity relationship (SAR) studies. Moreover, the use of subtype-selective radioligands is discussed." @default.
- W2382173 created "2016-06-24" @default.
- W2382173 creator A5056056907 @default.
- W2382173 creator A5060795115 @default.
- W2382173 creator A5081248127 @default.
- W2382173 date "2009-09-19" @default.
- W2382173 modified "2023-09-23" @default.
- W2382173 title "Dopamine Receptor Subtype-Selective Drugs: D2-Like Receptors" @default.
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