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- W2411070120 endingPage "54009" @default.
- W2411070120 startingPage "53997" @default.
- W2411070120 abstract "There is increasing interest in inhibitors targeting BET (bromodomain and extra-terminal) proteins because of the association between this family of proteins and cancer progression. BET inhibitors were initially shown to have efficacy in hematologic malignancies; however, a number of studies have now shown that BET inhibitors can also block progression of non-hematologic malignancies. In this Review, we summarize the efficacy of BET inhibitors in select solid tumors; evaluate the role of BET proteins in mediating resistance to current targeted therapies; and consider potential toxicities of BET inhibitors. We also evaluate recently characterized mechanisms of resistance to BET inhibitors; summarize ongoing clinical trials with these inhibitors; and discuss potential future roles of BET inhibitors in patients with solid tumors." @default.
- W2411070120 created "2016-06-24" @default.
- W2411070120 creator A5001372566 @default.
- W2411070120 creator A5039821839 @default.
- W2411070120 creator A5050914989 @default.
- W2411070120 creator A5076767039 @default.
- W2411070120 creator A5078031840 @default.
- W2411070120 date "2016-06-05" @default.
- W2411070120 modified "2023-10-14" @default.
- W2411070120 title "Targeting BET bromodomain proteins in solid tumors" @default.
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