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- W2414240129 abstract "Summary The radiochemical purity of the cobalt-57 complex of bleomycin could be enhanced by adjusting the pH of the final product to a value between 5 and 6. This radiopharmaceutical appeared to have better tumor visualizing properties compared to the not neutralized preparation. The clinical use of the cobalt-57 bleomycin complex is however limited by the long physical half-life of the label, causing a risk of radioactive contamination. It appeared to be possible to label bleomycin with radioactive cations (111In3+, 99mTc4+, 197Hg2+ and 67Cu2+) having suitable gamma ray energies and short half-lifes. These bleomycin complexes showed a high radiochemical purity judged by their behaviour on thin layer chromatography, paper chromatography, and electrophoresis, but their application as tumor visualizing radiopharmaceutical turned out to be disappointing compared with cobalt-57 bleomycin." @default.
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- W2414240129 date "1976-01-01" @default.
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- W2414240129 title "Labelling of Bleomycin with Cobalt-57, Indium-111, Technetium-99m, Mercury-197, Lead-203, and Copper-67" @default.
- W2414240129 doi "https://doi.org/10.1055/s-0038-1624940" @default.
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