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- W2479406918 endingPage "24" @default.
- W2479406918 startingPage "14" @default.
- W2479406918 abstract "Prostate cancer is initially responsive to androgen deprivation therapy, but most patients eventually develop castration-resistant disease. Enzalutamide is an androgen receptor (AR) inhibitor that targets several steps in the AR signaling pathway and has shown significant efficacy in the treatment of metastatic castration-resistant prostate cancer in patients with or without prior chemotherapy. To provide optimal treatment, it is important to understand the implications of enzalutamide use in the context of other therapies, as recent findings have suggested cross-resistance occurs between and within drug classes. Mutations and splice variants of AR also impact the course of prostate cancer. Future strategies involving enzalutamide should account for previous exposure to taxanes or antiandrogen therapies and the presence of AR variants that could affect efficacy." @default.
- W2479406918 created "2016-08-23" @default.
- W2479406918 creator A5004985848 @default.
- W2479406918 creator A5064376976 @default.
- W2479406918 date "2016-10-01" @default.
- W2479406918 modified "2023-10-17" @default.
- W2479406918 title "Treatment of metastatic castration-resistant prostate cancer (mCRPC) with enzalutamide" @default.
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